Triptorelin Acetate
Sequence:Pyr-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2
Appearance: White to off white powder
Standard: in-house
Application: Lab research
Supply Ability: 1000g per month
Purity: ≥98%
Payment: T/T, LC or DA
Delivery Time: Ready Stock in Local Warehouse, 1-3 days
Origin: China
Shipping: DHL, FedEx, TNT, EMS, By Sea, By Air
Can't sell to individuals
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Product Introduction
We supply Triptorelin Acetate
We offer Triptorelin Acetate, which is a synthetic analogue of gonadotropin- releasing hormone( GnRH) used in the treatment of advanced prostate cancer and unseasonable puberty. It works by dwindling the product of testosterone and estradiol, which can decelerate the growth of excrescences and delay the onset of puberty. Our product is of high chastity and is available in colorfulquantities.However, you can count on us to give you with high- quality products and excellent client service, If you're looking for dependable Triptorelin suppliers.
What's Triptorelin Acetate?
It is the acetate of triptorelin, with the active component triptorelin. Triptorelin is an instinctively synthesized and largely effective excipient analogue, which was first retailed in Germany in 1986. In order to ameliorate the bioavailability of general medicines, numerous mariners increase solubility and also enhance bioavailability. thus, the pharmacological goods and adverse responses of the two are harmonious. There are two lozenge forms of acetic acid triptorelin injection and sustained- release phrasings. Acetic acid triproline is a 5- Chemicalbook oxoprolyl- L- histidine L- tryptophan L- serine L- tyrosine- D- tryptophan L- leucoyl- L- arginyl- L- prolyl- L- glycinamide acetate, with a molecular formula of C64H82N18O13. XC2H4O2 and a molecular weight of1311.46. X60.02. According to computations without water or acetic acid, the content of C64H82N18O13 should be97.0% to103.0%.
Basic Information
Product Name: Triptorelin Acetate
Sequence:Pyr-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2<br>
CAS: 140194-24-7
MF: C64H82N18O13.C2H4O2
MW: 1371.52
EINECS: 194-124-7
MDL No.:MFCD28411371
Structural formula:
Origin: China
Application: Lab research
Delivery Time: in stock
Technical Specification
TEST |
SPECIFICATION |
RESULT |
Appearance |
White or almost white fluffy powder |
Conform |
Solubility |
Soluble in water |
Conform |
Water Content (Karl Fischer) |
≤ 8.0% |
4.8% |
Acetic Acid (By HPLC) |
≤ 15.0% |
9.8% |
Peptide Purity (By HPLC) |
≥ 98.0% |
99.76% |
Related Substance (By HPLC) |
Total Impurities(%) ≤ 2.0% |
0. 15% |
Largest Single Impurity(%) ≤ 1.0% |
0.04% |
|
Assay |
95.0 ~105.0% |
101.05% |
Conclusion |
This batch of product conforms with enterprise standard and qualified. |
Package 1g, 5g, 10g, 50g, 100g or according to your demands
Storage conditions 2- 8 ℃, dark, humidity- evidence, sealed and dry
Transportation conditions Transportation at room temperature
Shelf Life 24 months
Antitumor drugs
The active component of Triptorelin acetate is a synthetic analogue of gonadotropin- releasing hormone( GnRH), also known as tryptophan Rui Lin, DaFei Lin, Da Bi Jia, Gona Rui Lin. It's ananti-tumor medicine with pharmacological goods analogous to those of Gona Rui Lin and Bu Shen Rui Lin. Its structural enhancement is to replace the sixth L- glycine in the natural molecular structure with D- tryptophan, making its promoting effect more significant and the tube half- life longer, with advanced medicine efficacity. After intramuscular injection, the pituitary gland is originally stimulated to release luteinizing hormone( LH) and follicle stimulating hormone( FSH). When the pituitary gland enters the refractory period after long- term stimulation, the release of gonadotropins decreases, leading to a drop in coitus hormones to the position of castration. The below goods are reversible. Subcutaneous administration results in rapid-fire immersion, with a Tmax of 15 twinkles and maximum effect at 1 hour. Intramuscular injection of sustained- release phrasings can maintain efficacity for over 28 days. Clinically, it's substantially used for the treatment of endometriosis, hormone dependent prostate cancer, bone cancer, true unseasonable puberty in children, and supported reproductive technology.
Pharmacological action
The active component of acetic acid triptorelin is a synthetic analogue of gonadotropin- releasing hormone. Its structural revision involves replacing the sixth L- glycine in the natural molecular structure with D- tryptophan, making its synergistic effect more significant and tube half- life longer. After injection, the medicine originally stimulates the pituitary gland to release luteinizing hormone and chemotropin. later long- term stimulation, the pituitary gland enters an refractory period, and the release of gonadotropins decreases, leading to a drop in coitus steroids to the position of castration. The below goods are reversible. Subcutaneous administration results in rapid-fire immersion, with tube attention reaching its peak at 15- 60 twinkles and maximum effect at 1 hour. Intramuscular injection of sustained- release phrasings can maintain efficacity for over 28 days.
Application
it is a synthetic peptide hormone analogue that's used in the treatment of colorful hormone-dependent conditions similar as prostate cancer, endometriosis, and uterine fibroids. It belongs to the class of gonadotropin- releasing hormone( GnRH) agonists, which work by suppressing the product of certain hormones in the body.
In the treatment of prostate cancer, it is used to reduce the situations of testosterone in the body. This is because prostate cancer cells bear testosterone to grow and divide, and reducing its product can help decelerate down or indeed stop the growth of the cancer. It's generally given as an injection every one to six months.
In the treatment of endometriosis and uterine fibroids, it is used to temporarily suppress the product of estrogen in the body. This can help to palliate symptoms similar as pelvic pain, heavy bleeding, and gravidity. It's generally given as an injection every one to three months.
it is a veritably potent drug and should only be used under the supervision of a healthcare provider. It may beget side goods similar as hot flashes, night sweats, headaches, and mood changes. It may also increase the threat of developing osteoporosis, so regular bone viscosity tests may be necessary.
In conclusion, it is a effective drug that's used in the treatment of colorful hormone-dependent conditions. It works by suppressing the product of certain hormones in the body, and is generally given as an injection every one to six months. still, it should only be used under the supervision of a healthcare provider due to its energy and implicit side goods.
Packing & Shipping
Packing:1kg/foil bag;5kg/carton;25kg/fiber drum;or packing as your request.
Customization:Customized logo; Customized packaging; Graphic customization
Shipping:
Item |
Quantity |
ETA time |
Shipping Method |
By Courier |
≤50kg |
7-15days |
Fedex, DHL,UPS,TNT,EMS ect. Fast and convenient |
By Air |
50kg~200kg |
3-5days |
Fast and cheap |
By Sea |
Large quantity |
20-35days |
Cheapest way |
Payment Term
Why Choose Xi'an Yihui?
Customer feedback
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Our advantage
Rich experice: we have 13 Years professional experience;
Customers all over the word: sell to more than 100 countries;
Provide diversified products: the products have been applied to all major international brands in the fields of drugs, dietary supplements, cosmetics, animal nutrition and functional food.
Price advance: low MOQ with competitive price;
Quality certification: ISO; Halal; Kosher certified
After-sales service: Professional team 7*24 hours customer service.
Contact Yihui company
In summary, as a professional Triptorelin acetatemanufacturer, we have advanced technology, scale advantage, the best quality, rich production experience, and excellent services. These advantages will make it stand out in the market competition and win more customer trust and support. if you need it, pls feel free to contact us any time. we will reply you asap.
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Tel: 0086-29-89695240
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